The synthesis of bicyclic 1,2,3,4-tetrahydro-1,4-benzodiazepin-5-ones from 2-(o-nitrobenzyl)-1,2-thiazine-1-oxide precursors

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1. B.E. Evans, K.E. Rittle, M.G. Bock, R.M. DiPardo, R.M. Freidinger, W.L. Whitter, G.F. Lundell, D.F. Veber, P.S. Anderson, R.S.L. Chang, V.J. Lotti, D.J. Cerino, T.B. Chen, P.J. Kling, K.A. Kunkel, J.P. Springer and J. Hirschfield. J. Med. Chem. 31 (1988), p. 2235. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
A.A. Patchett and R.P. Nargund. Annu. Rep. Med. Chem. 35 (2000), p. 289.
S. Herrero, M.T. García-López and R. Herranz. J. Org. Chem. 68 (2003), p. 4582. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

2. See, for example: (a) L.H. Sternbach. J. Med. Chem. 22 (1979), p. 1. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
L.H. Sternbach. Prog. Drug. Res. 22 (1978), p. 229. View Record in Scopus | Cited By in Scopus
G.A. Showell, S. Bourrain, J.G. Neduvelil, S.R. Fletcher, R. Baker, A.P. Watt, A.E. Fletcher, S.B. Freedman, J.A. Kemp, G.R. Marshall, S. Patel, A.J. Smith and V.G. Matassa. J. Med. Chem. 37 (1994), p. 719. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
B.A. Bunin, M.J. Plunkett and J.A. Ellman. Proc. Natl. Acad. Sci. USA 91 (1994), p. 4708. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

3. See, for example: (a) W.B. Wright, H.J. Brabander, E.N. Greenblatt, I.P. Day and R.A. Hardy. J. Med. Chem. 21 (1978), p. 1087. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
C.G. Boojamra, K.M. Burow, L.A. Thompson and J.A. Ellman. J. Org. Chem. 62 (1997), p. 1240. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
T.A. Keating and R.W. Armstrong. J. Org. Chem. 61 (1996), p. 8935. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
R.R. Webb, P.R. Barker, M. Baier, M.E. Reynolds, K.D. Robarge, B.K. Blackburn, M.H. Tichler and K.J. Weese. Tetrahedron Lett. 35 (1994), p. 2113. Abstract | Abstract + References | PDF (283 K) | View Record in Scopus | Cited By in Scopus

4. D.E. Thurston and D.S. Bose. Chem. Rev. 94 (1994), p. 433. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
P. Molina, I. Díaz and A. Tárraga. Tetrahedron 51 (1995), p. 5617. Abstract | Abstract + References | PDF (806 K) | View Record in Scopus | Cited By in Scopus
I.A. O'Neil, S. Thompson, C.L. Murray and S.B. Kalindjian. Tetrahedron Lett. 39 (1998), p. 7787. SummaryPlus | Full Text + Links | PDF (201 K) | View Record in Scopus | Cited By in Scopus
N. Cooper, D.R. Hagan, A. Tiberghien, T. Ademefun, C.S. Matthews, P.W. Howard and D.E. Thurston. Chem. Commun. (2002), p. 1784.

5. T. Sugimori, T. Okawa, S. Eguchi, A. Kakehi, E. Yashima and Y. Okamoto. Tetrahedron 54 (1998), p. 7997. Abstract | Abstract + References | PDF (712 K) | View Record in Scopus | Cited By in Scopus
A. Witt and J. Bergman. J. Org. Chem. 66 (2001), p. 2784. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

6. M. Artico, R. Silvestri, E. Pagnozzi, G. Stefancich, S. Massa, A.G. Loi, M. Putzolu, S. Corrias, M.G. Spiga and P. La Colla. Bioorg. Med. Chem. 4 (1996), p. 837 and references cited therein . Abstract | Abstract + References | PDF (1353 K) | View Record in Scopus | Cited By in Scopus

7. F. Novelli, A. Sparatore, B. Tass and F. Sparatore. Bioorg. Med. Chem. Lett. 9 (1999), p. 3031 and references cited therein . Abstract | Abstract + References | PDF (231 K) | View Record in Scopus | Cited By in Scopus

8. W. Fröstl and L. Maître. Pharmacopsych. 22 (1989), p. 54. View Record in Scopus | Cited By in Scopus
G. Broggini, G. Molteni, A. Terraneo and G. Zecchi. Tetrahedron 55 (1999), p. 14803. Abstract | Abstract + References | PDF (263 K) | View Record in Scopus | Cited By in Scopus

9. G. Gründer, T. Siessmeier, C. Lange-Asschenfeldt, I. Vernaleken, H.-G. Buchholz, P. Stoeter, A. Drzezga, H. Lüddens, F. Rösch and P. Bartenstein. Eur. J. Nucl. Med. 28 (2001), p. 1463. View Record in Scopus | Cited By in Scopus

10. A. Walser and R.I. Fryer. In: E.C. Taylor and A. Weissberger, Editors, Chemistry of heterocyclic compoundsBicyclic diazepines Vol. 50, Wiley, Chichester, UK (1991), p. 431 Chapters V–VIII .

11. K. Meguro and Y. Kuwada. Tetrahedron Lett. 10 (1970), p. 4039. Abstract | Abstract + References | PDF (176 K)
G. Mohiuddin, P.S. Reddy, K. Ahmed and C.V. Ratnam. Heterocycles 24 (1986), p. 3489.
Santilli, A. A.; Osdene, T. S. U.S. Patent 3,336,330, 1967; Chem. Abstr. 68, 21972.
Hester, J. B. U.S. Patent 3,896,109, 1975; Chem. Abstr. 84, 17440.
A.N. Osman, A.A. El-Gendy, R.H. Omar, L. Wagdy and A.H. Omar. Ind. J. Chem. (B) 41B (2002), p. 871. View Record in Scopus | Cited By in Scopus

12. Santilli, A. A.; Osdene, T. S. U.S. Patent 3,457,258; Chem. Abstr. 1969, 71, 101898.

13. J.B. Hester, A.D. Rudzik and B.V. Kamadar. J. Med. Chem. 14 (1971), p. 1078. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

14. T. Kaneko, H. Wong, T.W. Doyle, W.C. Rose and W.T. Bradner. J. Med. Chem. 28 (1985), p. 388. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

15. R.M. Keenan, J.F. Callahan, J.M. Samanen, W.E. Bondinell, R.R. Calvo, L. Chen, C. DeBrosse, D.S. Eggleston, R.C. Haltiwanger, S.M. Hwang, D.R. Jakas, T.W. Ku, W.H. Miller, K.A. Newlander, A. Nichols, M.F. Parker, L.S. Southhall, I. Uzinskas, J.A. Vasko-Moser, J.W. Venslavsky, A.S. Wong and W.F. Huffman. J. Med. Chem. 42 (1999), p. 545. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

16. A.A. Santilli and T.S. Osdene. J. Org. Chem. 30 (1965), p. 2100. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
N. Matsunaga, H. Harada, T. Aoyama and T. Shioiri. Heterocycles 33 1 (1992), p. 235.

17. M. Miyamoto, S. Kondo, H. Naganawa, K. Maeda, M. Ohno and H. Umezawa. J. Antibiot. 30 (1977), p. 340.
K.-H. Weber. Arch. Pharmaz. 302 (1969), p. 584. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

18. V. Santagada, E. Perissutti, F. Fiorino, B. Vivenzio and G. Caliendo. Tetrahedron Lett. 42 (2001), p. 2397. SummaryPlus | Full Text + Links | PDF (62 K) | View Record in Scopus | Cited By in Scopus
G. Molteni, G. Broggini and T. Pilati. Tetrahedron: Asymmetry 13 (2002), p. 2491. SummaryPlus | Full Text + Links | PDF (255 K) | View Record in Scopus | Cited By in Scopus

19. B. Anwar, P. Grimsey, K. Hemming, M. Krajniewski and C. Loukou. Tetrahedron Lett. 41 (2000), p. 10107. SummaryPlus | Full Text + Links | PDF (66 K) | View Record in Scopus | Cited By in Scopus
S. Eguchi, K. Yamashita and Y. Matsushita. Synlett (1992), p. 295. Full Text via CrossRef

20. J.D. White, W.E. Haefliger and M.J. Dimsdale. Tetrahedron 26 (1970), p. 233. Abstract | Abstract + References | PDF (857 K) Abstract | Abstract + References | PDF (857 K) | View Record in Scopus | Cited By in Scopus

21. M.D. Surman, M.J. Mulvihill and M.J. Miller. Org. Lett. 4 (2002), p. 139. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

22. M. Julia, N. Hurion and D.T. Huynh. Chimica Therapeutica 5 (1970), p. 343.

23. A. Pedrazzoli, L. Dall'Asta and P. Ferrario. Bull. Soc. Chim. France (1968), p. 407.

24. T. Wang, A.S. Lui and I.S. Cloudsdale. Org. Lett. 1 (1999), p. 1835. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

25. F. Ammadi, S. Boukhris, A. Souizi and G. Coudert. Tetrahedron Lett. 40 (1999), p. 6517. SummaryPlus | Full Text + Links | PDF (126 K) | View Record in Scopus | Cited By in Scopus

26. Yoo, H. W.; Lee, J. W.; Suh, M. E. Yakhak Hoechi 1989 33, 246; Chem. Abstr. 112, 216885.

27. C. Corral, R. Madroñero and S. Vega. J. Heterocycl. Chem. 14 (1977), p. 99. View Record in Scopus | Cited By in Scopus

28. L. Abrous, J. Hynes, Jr., S.R. Friederich, A.B. Smith, III and R. Hirschmann. Org. Lett. 3 (2001), p. 1089. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

29. A. Bauer and K.-H. Weber. Z. Naturforsch. 29b (1974), p. 670. View Record in Scopus | Cited By in Scopus

30. D.E. Thurston, P.T.P. Kaumaya and L.H. Hurley. Tetrahedron Lett. 25 (1984), p. 4706.

31. K.H. Wünsch, K.H. Stahnke and P. Gomoll. Z. Chem. 10 (1970), p. 219.
P.I. Ittyerah and F.G. Mann. J. Chem. Soc. (1958), p. 467. Full Text via CrossRef
D. Misiti, F. Gatta and R. Landi-Vittory. J. Heterocycl. Chem. 8 (1971), p. 231.
G.L. Grunewald, V.H. Dahanukar, P. Ching and K.R. Criscione. J. Med. Chem. 39 (1996), p. 3539. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

32. G.F. Field, W.J. Zally and L.H. Sternbach. J. Org. Chem. 36 (1971), p. 777. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus
Y. Yamada, T. Oine and I. Inoue. Bull. Chem. Soc. Jpn 47 2 (1974), p. 339. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

33. F. Hollywood, Z.U. Khan, E.F.V. Scriven, R.K. Smalley, H. Suschitzky, D.R. Thomas and R. Hull. J. Chem. Soc., Perkin Trans. 1 (1982), p. 431. Full Text via CrossRef

34. S.M. Weinreb. Acc. Chem. Res. 21 (1988), p. 313. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus

35. R. Bussas, G. Kresze, H. Münsterer and A. Schwöbel. Sulfur Rep. 2 (1983), p. 215.

36. D.A. Evans and G.C. Andrews. Acc. Chem. Res. 7 (1974), p. 147. Full Text via CrossRef | View Record in Scopus | Cited By in Scopus